SCHEMBL7380728

SCHEMBL7380728

Cc1c(CCN)[nH]c2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.55
MAPK1 P28482 2/20 0.55
NPSR1 Q6W5P4 1/20 0.55
AHR P35869 1/20 0.52
HTR6 P50406 6/20 0.49
RAB9A P51151 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
HTR1D P28221 2/20 0.44
HTR7 P34969 2/20 0.44
MPO P05164 1/20 0.44
CYP2A6 P11509 1/20 0.44
NFKB1 P19838 1/20 0.44
HTR1B P28222 1/20 0.44
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
CTSK P43235 1/20 0.44
CYP2A13 Q16696 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30952639 1.00 MAPT (0.55) MAPTMAPK1NPSR1AHRHTR6
SCHEMBL6953567 0.85 AHR (0.55) MAPTMAPK1NPSR1AHRHTR6
SCHEMBL12808068 0.83 RAB9A (0.60) MAPTMAPK1NPSR1AHRHTR6
SCHEMBL31405650 0.81 ALDH1A1 (0.59) MAPTMAPK1NPSR1AHRHTR6
SCHEMBL13485647 0.80 AHR (0.59) MAPTAHRRAB9ACYP1A2CYP3A4
SCHEMBL10082865 0.80 RAB9A (0.57) MAPTAHRRAB9ACYP1A2CYP3A4
SCHEMBL24405131 0.79 HTR6 (0.66) MAPTAHRHTR6RAB9AL3MBTL1
SCHEMBL6330362 0.79 OXER1 (0.56) MAPTAHRRAB9ACYP1A2CYP3A4
SCHEMBL3886866 0.79 HTR6 (0.63) MAPTMAPK1NPSR1HTR6CYP1A2
SCHEMBL7847012 0.79 KDM4E (0.63) MAPTMAPK1NPSR1AHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118255830-A S1PR2 modulators and uses thereof 北京昌平实验室 2024-06-28 CN disclosed
EP-0420086-B1 Pyrimidoindole derivatives and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO (JP) 1995-12-13 EP disclosed
US-5256780-A Serotonin antagonist FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-10-26 US disclosed
US-5180728-A Antagonists of 5-hydroxytryptamine FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1993-01-19 US disclosed
EP-0420086-A2 Pyrimidoindole derivatives and processes for preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-04-03 EP disclosed