SCHEMBL7380790

SCHEMBL7380790

Cc1ccc([N+](=O)[O-])cc1C(=O)NC(CO)Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.52
SMN1; SMN2 Q16637 3/20 0.50
NPC1 O15118 1/20 0.50
TP53 P04637 1/20 0.50
RAB9A P51151 1/20 0.50
MAPK1 P28482 3/20 0.47
CYP3A4 P08684 2/20 0.47
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
ROCK2 O75116 3/20 0.46
ROCK1 Q13464 3/20 0.46
RPS6KA5 O75582 2/20 0.46
RPS6KA4 O75676 2/20 0.46
PRKACA P17612 2/20 0.46
GSK3B P49841 2/20 0.46
PRKX P51817 2/20 0.46
PRKG1 Q13976 2/20 0.46
CLK4 Q9HAZ1 2/20 0.46
LIMK1 P53667 1/20 0.46
ALDH1A1 P00352 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789861 1.00 LMNA (0.52) LMNASMN1; SMN2NPC1TP53RAB9A
SCHEMBL7383243 0.81 MAPK1 (0.51) NPC1RAB9AMAPK1CYP3A4KMT2A
SCHEMBL7376752 0.81 MAPK1 (0.51) NPC1RAB9AMAPK1CYP3A4KMT2A
SCHEMBL7382779 0.81 ALDH1A1 (0.64) LMNASMN1; SMN2NPC1TP53RAB9A
SCHEMBL7786734 0.81 NPC1 (0.70) LMNASMN1; SMN2NPC1TP53RAB9A
SCHEMBL7381190 0.81 NPC1 (0.70) LMNASMN1; SMN2NPC1TP53RAB9A
SCHEMBL7782237 0.80 CAPN1 (0.49) LMNASMN1; SMN2NPC1TP53RAB9A
SCHEMBL7782235 0.80 CAPN1 (0.49) LMNASMN1; SMN2NPC1TP53RAB9A
SCHEMBL29018285 0.78 CTSD (0.55) LMNASMN1; SMN2MAPK1CYP3A4KMT2A
SCHEMBL29018283 0.78 CTSD (0.55) LMNASMN1; SMN2MAPK1CYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed
EP-0944584-A1 BENZAMIDOALDEHYDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-09-29 EP disclosed
WO-1998023581-A1 BENZAMIDOALDEHYDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-06-04 WO disclosed