SCHEMBL7381815

SCHEMBL7381815

CC12CC[C@](C(=O)N3CCC4(C=Cc5ccccc54)CC3)(OC1=O)C2(C)C

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.58
POLB P06746 1/20 0.58
ALDH1A1 P00352 3/20 0.58
NPSR1 Q6W5P4 2/20 0.58
LMNA P02545 1/20 0.58
HTT P42858 1/20 0.58
HSD11B1 P28845 1/20 0.50
NR1H2 P55055 1/20 0.47
NR1H3 Q13133 1/20 0.47
PTBP1 P26599 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7381813 1.00 GAA (0.58) GAAPOLBALDH1A1NPSR1LMNA
SCHEMBL395086 0.74 HSD11B1 (0.64) HSD11B1NR1H2NR1H3
SCHEMBL3455531 0.73 GAA (0.60) GAAPOLBALDH1A1NPSR1LMNA
SCHEMBL12204828 0.72 POLB (0.74) GAAPOLBALDH1A1NPSR1LMNA
SCHEMBL766158 0.71 ALDH1A1 (0.60) GAAPOLBALDH1A1NPSR1LMNA
SCHEMBL1577378 0.69 HSD11B1 (0.57) HSD11B1NR1H2NR1H3
SCHEMBL1577665 0.69 HSD11B1 (0.54) HSD11B1NR1H2NR1H3
SCHEMBL30107924 0.69 HSD11B1 (0.54) HSD11B1NR1H2NR1H3
SCHEMBL8472020 0.67 OXTR (0.57) HSD11B1
SCHEMBL3457632 0.67 LMNA (0.61) GAAPOLBALDH1A1NPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0450761-A1 Spirocyclic oxytocin antagonists MERCK & CO. INC. (US) 1991-10-09 EP claimed