SCHEMBL7382016

SCHEMBL7382016

Cc1cccc(CC(Cc2cccc(C)c2C)C(=O)O)c1C

nearest known ligand 0.81

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.48
CYP1A2 P05177 1/20 0.47
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
PPARA Q07869 2/20 0.40
NR3C1 P04150 1/20 0.40
PGR P06401 1/20 0.40
NR3C2 P08235 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
PTGES O14684 1/20 0.40
ALOX5 P09917 1/20 0.40
LMNA P02545 1/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
FOLH1 Q04609 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GLA P06280 1/20 0.39
STING1 Q86WV6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8053590 0.87 KMT2A (0.50) PPARGCYP1A2ALDH1A1HPGDPPARA
SCHEMBL7384644 0.85 PPARG (0.57) PPARGCYP1A2ALDH1A1HPGDPPARA
SCHEMBL24899379 0.84 L3MBTL1 (0.46) PPARGPPARANR3C1PGRNR3C2
SCHEMBL430339 0.84 L3MBTL1 (0.46) PPARGPPARANR3C1PGRNR3C2
SCHEMBL30013065 0.82 NOS3 (0.53) ALDH1A1HPGDLMNAL3MBTL1
SCHEMBL9188703 0.82 NOS3 (0.53) ALDH1A1HPGDLMNAL3MBTL1
SCHEMBL14246987 0.82 PPARG (0.41) PPARGALDH1A1HPGDPPARANR3C1
SCHEMBL5326602 0.82 NOS3 (0.53) ALDH1A1HPGDLMNAL3MBTL1
SCHEMBL34461657 0.82 NOS3 (0.53) ALDH1A1HPGDLMNAL3MBTL1
SCHEMBL5145689 0.82 PPARG (0.43) PPARGCYP1A2PPARANR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610177-A Acylated amino acids as endothelin antagonists WARNER-LAMBERT COMPANY (US) 1997-03-11 US disclosed
US-4870183-A RENIN INHIBITORS, HYPOTENSIVES KISSEI PHARMACEUTICAL CO., LTD. (JP) 1989-09-26 US disclosed
EP-0252727-A1 Novel amino acid derivatives Kissei Pharmaceutical Co. Ltd. (JP) 1988-01-13 EP disclosed