SCHEMBL7382104

SCHEMBL7382104

COc1cc2cc(C(=O)O)oc(=O)c2cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.50
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 4/20 0.43
POLB P06746 1/20 0.43
ALDH1A1 P00352 3/20 0.42
ELANE P08246 3/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA2 P00918 1/20 0.41
CA3 P07451 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA14 Q9ULX7 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
HTT P42858 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766674 0.80 PIM1 (0.55) PIM1KMT2AKDM4EALDH1A1CA12
SCHEMBL9319353 0.76 BCL2L1 (0.46) PIM1KMT2AKDM4EPOLBCA12
SCHEMBL5560761 0.74 KDM4E (0.64) KMT2ASMN1; SMN2KDM4EPOLBALDH1A1
SCHEMBL11845147 0.74 CA12 (0.55) PIM1KMT2ASMN1; SMN2KDM4EPOLB
SCHEMBL10712556 0.73 HPGD (0.50) PIM1KDM4EPOLBALDH1A1CA12
SCHEMBL7470487 0.71 PIM1 (0.61) PIM1KMT2ASMN1; SMN2KDM4EPOLB
SCHEMBL11745931 0.71 PIM1 (0.57) PIM1KMT2ASMN1; SMN2KDM4EPOLB
SCHEMBL31064944 0.70 ALDH1A1 (0.56) PIM1SMN1; SMN2KDM4EPOLBALDH1A1
SCHEMBL20563607 0.70 PIM1 (0.56) PIM1KDM4EALDH1A1LMNATP53
SCHEMBL175987 0.69 ALDH1A1 (0.59) PIM1KMT2ASMN1; SMN2KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6486155-B1 Method of inhibiting neoplastic cells with isoquinoline derivatives CELL PATHWAYS INC 2002-11-26 US disclosed
WO-1998038168-A1 ISOQUINOLINONE DERIVATIVES, PROCESS FOR PREPARING THE SAME, AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS TANABE SEIYAKU CO., LTD. (JP) 1998-09-03 WO disclosed
US-5371220-A Bicyclo-heterocyclic intermediates for cephalosporin compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-12-06 US disclosed
US-5232918-A Bactericides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-08-03 US disclosed
US-5019570-A Antibioics IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-05-28 US disclosed