SCHEMBL7385487

SCHEMBL7385487

c1ccc2[nH]c(C3CNCCN3)cc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.41
AOC3 Q16853 2/20 0.38
MAOB P27338 1/20 0.37
HRH4 Q9H3N8 2/20 0.36
HRH3 Q9Y5N1 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
LOXL2 Q9Y4K0 1/20 0.35
FLT3 P36888 1/20 0.35
CYP2A6 P11509 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA3 P07451 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA13 Q8N1Q1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3330972 0.79 NR1H4 (0.41) PARP1AOC3MAOB
SCHEMBL5382942 0.77 METTL3 (0.43) PARP1AOC3MAOBCYP2A6
SCHEMBL2467564 0.73 HTR2A (0.49) PARP1
SCHEMBL9704857 0.72 DRD2 (0.50)
SCHEMBL29688552 0.71 MAOB (0.49) AOC3MAOBHRH4HRH3MAPT
SCHEMBL1237690 0.71 MAOB (0.49) AOC3MAOBHRH4HRH3MAPT
SCHEMBL7866443 0.71 CHRNB2 (0.41) AOC3NPC1RAB9ALOXL2FLT3
SCHEMBL4559567 0.71 HDAC8 (0.48) HRH4HRH3LOXL2
SCHEMBL1637550 0.70 SLC6A2 (0.49) MAOBKDM4E
SCHEMBL2243349 0.70 PARP1 (0.55) PARP1AOC3NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0648766-A1 AGENT ACTING ON THE CENTRAL NERVOUS SYSTEM, METHOD FOR ITS PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH AGENT VITA-INVEST, S.A. (ES) 1995-04-19 EP disclosed
WO-1994025454-A1 AGENT ACTING ON THE CENTRAL NERVOUS SYSTEM, METHOD FOR ITS PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH AGENT VITA-INVEST, S.A. (ES) 1994-11-10 WO disclosed