SCHEMBL7386284

SCHEMBL7386284

ClCCNCc1cncc(-c2ccccc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
FDPS P14324 2/20 0.44
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HTR1A P08908 1/20 0.40
CNR1 P21554 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SCN2A Q99250 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.39
HDAC1 Q13547 1/20 0.38
CHRM2 P08172 1/20 0.37
SCN8A Q9UQD0 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
MAOA P21397 1/20 0.37
KDM4C Q9H3R0 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7397089 0.91 CYP11B1 (0.47) CYP11B1CYP11B2FDPSMEN1KMT2A
SCHEMBL7385522 0.90 CYP11B1 (0.46) CYP11B1CYP11B2FDPSCHRM2SCN8A
SCHEMBL7395929 0.85 HTR1A (0.48) CYP11B1CYP11B2HTR1ACHRM2CYP1A2
SCHEMBL7392006 0.80 DRD4 (0.60) CYP11B1CYP11B2HTR1AHDAC1
SCHEMBL2646363 0.78 CYP11B1 (0.54) CYP11B1CYP11B2FDPSCNR1SCN2A
SCHEMBL7391666 0.77 DRD4 (0.50) CYP11B1CYP11B2SCN8AMAOA
SCHEMBL7396125 0.77 DRD4 (0.53) CNR1SCN2ASCN10A
SCHEMBL7395367 0.77 DRD4 (0.50) MEN1KMT2AHTR1A
SCHEMBL29373657 0.77 FDPS (0.53) CYP11B1CYP11B2FDPSCNR1SCN2A
SCHEMBL8625517 0.77 PRMT6 (0.57) CYP11B1CYP11B2FDPSATMCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1246319-C Amino (thio) ether derivative MERCK PATENT AG (DE) 2006-03-22 CN disclosed
EP-1123933-A1 2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]chromane as CNS active agent MERCK PATENT GmbH (DE) 2001-08-16 EP disclosed
US-5767132-A CENTRAL NERVOUS SYSTEM MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-06-16 US disclosed
CN-1130180-A Amino (thio) ether derivative MERCK PATENT AG (DE) 1996-09-04 CN disclosed
EP-0707007-A1 Amino(thio)ether derivatives as CNS active agents MERCK PATENT GmbH (DE) 1996-04-17 EP disclosed