SCHEMBL7386450

SCHEMBL7386450

CC(=O)OC(=O)[C@@H]1CN(C(=O)N(c2ccccc2)c2ccccc2)CCN1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 1/20 0.47
ALDH1A1 P00352 5/20 0.41
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KMT2A Q03164 2/20 0.40
TACR1 P25103 3/20 0.39
CHRM4 P08173 2/20 0.39
CHRM3 P20309 2/20 0.39
MEN1 O00255 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL7386447 0.85 AGTR2 (0.54) AGTR2ALDH1A1POLBSMN1; SMN2L3MBTL1
Acetic Acid SCHEMBL7386453 0.85 AGTR2 (0.54) AGTR2ALDH1A1POLBSMN1; SMN2L3MBTL1
SCHEMBL30451454 0.83 AGTR2 (0.58) AGTR2ALDH1A1POLBSMN1; SMN2L3MBTL1
SCHEMBL30743851 0.81 AGTR2 (0.52) AGTR2ALDH1A1POLBSMN1; SMN2L3MBTL1
SCHEMBL7387158 0.71 AGTR2 (0.47) AGTR2ALDH1A1TACR1CHRM4CHRM3
SCHEMBL7391886 0.71 AGTR2 (0.47) AGTR2ALDH1A1TACR1CHRM4CHRM3
SCHEMBL10281640 0.71 TSHR (0.48) ALDH1A1SMN1; SMN2KMT2ACHRM4CHRM3
SCHEMBL7388960 0.70 ALDH1A1 (0.61) AGTR2ALDH1A1POLBSMN1; SMN2L3MBTL1
SCHEMBL7656754 0.69 SIGMAR1 (0.51) ALDH1A1KMT2AMEN1
SCHEMBL7467929 0.68 ALDH1A1 (0.77) AGTR2ALDH1A1POLBSMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995000498-A1 N,N-DIACYLPIPERAZINES MERCK & CO., INC. (US) 1995-01-05 WO disclosed
US-5348955-A Angiotensis II antagonists MERCK & CO., INC. (US) 1994-09-20 US disclosed
US-5292726-A N,N-diacylpiperazines MERCK & CO., INC. (US) 1994-03-08 US disclosed
WO-1992020661-A1 N, N-DIACYLPIPERAZINES MERCK & CO., INC. (US) 1992-11-26 WO disclosed