SCHEMBL738862

SCHEMBL738862

Nc1cccc(CCN2CCOCC2)c1N

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.47
POLB P06746 1/20 0.45
CYP2A13 Q16696 5/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
ATM Q13315 1/20 0.41
CXCR4 P61073 1/20 0.40
KCNH2 Q12809 1/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.40
NCF1 P14598 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30115041 0.91 SIGMAR1 (0.54) SIGMAR1POLBCYP2A13L3MBTL1CNR1
SCHEMBL3718831 0.87 SIGMAR1 (0.60) SIGMAR1POLBCYP2A13L3MBTL1HRH3
SCHEMBL2327709 0.85 HRH3 (0.59) SIGMAR1L3MBTL1HRH3KCNH2
SCHEMBL6055273 0.83 CYP2A13 (0.57) CYP2A13HRH3CXCR4NCF1
SCHEMBL31172442 0.83 CYP2A13 (0.57) CYP2A13HRH3CXCR4NCF1
SCHEMBL28344098 0.81 SIGMAR1 (0.49) SIGMAR1POLBCYP2A13CNR1CNR2
SCHEMBL18108811 0.80 PARP1 (0.53) CNR1CNR2
SCHEMBL6526231 0.79 POLB (0.47) SIGMAR1POLB
SCHEMBL22716816 0.78 L3MBTL3 (0.39) SIGMAR1L3MBTL1HRH3KCNH2
SCHEMBL5323909 0.77 HRH3 (0.54) SIGMAR1POLBCYP2A13L3MBTL1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113924296-A 1,3, 4-oxadiazole derivative compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions comprising the same 株式会社钟根堂 2022-01-11 CN disclosed
CN-105189481-A Pyridine cdk9 kinase inhibitors ABBVIE INC 2015-12-23 CN disclosed
US-8138177-B2 Benzimidazolone derivatives as CB2 receptor ligands PFIZER INC. (US) 2012-03-20 US disclosed
EP-1318978-B1 N-ACYLSULFONAMIDE APOPTOSIS PROMOTERS ABBOTT LAB (US) 2006-02-08 EP disclosed
US-5716953-A MODIFIERS OF GASTRIN AND CHOLECYSTOKININS GLAXO WELLCOME S.P.A. (IT) 1998-02-10 US disclosed