SCHEMBL739438

SCHEMBL739438

CCOC(=O)C1=C(Cl)c2sc3c(c2CN1C)CCCC3

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.47
KDM4E B2RXH2 6/20 0.47
MAPT P10636 6/20 0.47
GAA P10253 4/20 0.47
HSD17B10 Q99714 3/20 0.47
HPGD P15428 3/20 0.47
ALOX15 P16050 2/20 0.47
MAPK1 P28482 1/20 0.47
TLR2 O60603 5/20 0.43
ADRA2A P08913 2/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
KMT2A Q03164 1/20 0.41
TSHR P16473 4/20 0.41
NPSR1 Q6W5P4 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
TLR1 Q15399 1/20 0.40
LMNA P02545 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741438 0.86 ALDH1A1 (0.47) ALDH1A1KDM4EMAPTGAAHSD17B10
SCHEMBL739356 0.76 ALDH1A1 (0.37) ALDH1A1KDM4EMAPTGAAHSD17B10
SCHEMBL741117 0.73 ALDH1A1 (0.36) ALDH1A1KDM4EMAPTGAAHSD17B10
SCHEMBL3477086 0.69 ALDH1A1 (0.37) ALDH1A1KDM4EMAPTGAAHSD17B10
SCHEMBL10241785 0.68 MAPT (0.75) ALDH1A1KDM4EMAPTGAAHSD17B10
SCHEMBL14926951 0.67 ALDH1A1 (0.40) ALDH1A1KDM4EMAPTGAAHSD17B10
SCHEMBL19879527 0.65 MAPT (0.69) ALDH1A1KDM4EMAPTGAAHSD17B10
SCHEMBL19141297 0.65 MAPT (0.69) ALDH1A1KDM4EMAPTGAAHSD17B10
SCHEMBL6999008 0.65 ALDH1A1 (0.69) ALDH1A1KDM4EMAPTGAAHSD17B10
SCHEMBL29373525 0.65 MAPT (0.57) ALDH1A1KDM4EMAPTGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430029-A1 THIENO [2, 3-B]PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS Katholieke Universiteit Leuven (BE) 2012-03-21 EP disclosed
WO-2010130842-A1 THIENO [2, 3-B] PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2010-11-18 WO disclosed