SCHEMBL739356

SCHEMBL739356

CCOC(C(=O)OC)C1=C(Cl)c2sc3c(c2CN1C)CCCC3

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.37
MAPT P10636 7/20 0.37
KDM4E B2RXH2 4/20 0.37
GAA P10253 4/20 0.37
ALOX15 P16050 4/20 0.37
HSD17B10 Q99714 4/20 0.37
HPGD P15428 2/20 0.37
MAPK1 P28482 2/20 0.37
TSHR P16473 4/20 0.37
TLR2 O60603 4/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
LMNA P02545 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
KMT2A Q03164 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741117 0.84 ALDH1A1 (0.36) ALDH1A1MAPTKDM4EGAAALOX15
SCHEMBL739438 0.76 ALDH1A1 (0.47) ALDH1A1MAPTKDM4EGAAALOX15
SCHEMBL741438 0.67 ALDH1A1 (0.47) ALDH1A1MAPTKDM4EGAAALOX15
SCHEMBL134946 0.67 KDM4E (0.48) ALDH1A1KDM4EGAAHSD17B10HPGD
SCHEMBL739355 0.65
SCHEMBL14926951 0.63 ALDH1A1 (0.40) ALDH1A1MAPTKDM4EGAAHSD17B10
SCHEMBL740648 0.61 SLC22A12 (0.41) KDM4ESMN1; SMN2KMT2ATP53
SCHEMBL3477086 0.60 ALDH1A1 (0.37) ALDH1A1MAPTKDM4EGAAHSD17B10
SCHEMBL10241785 0.58 MAPT (0.75) ALDH1A1MAPTKDM4EGAAALOX15
SCHEMBL22074117 0.57 ALDH1A1 (0.38) ALDH1A1MAPTKDM4EGAAALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430029-A1 THIENO [2, 3-B]PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS Katholieke Universiteit Leuven (BE) 2012-03-21 EP disclosed
WO-2010130842-A1 THIENO [2, 3-B] PYRIDINE DERIVATIVES AS VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2010-11-18 WO disclosed