SCHEMBL7397667

SCHEMBL7397667

O=[N+]([O-])c1ccc2[nH]c3c(c2c1)CCNc1ccc(Br)cc1-3

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 13/20 0.69
CDK5 Q00535 12/20 0.69
CDK5R1 Q15078 12/20 0.69
CCNB2 O95067 12/20 0.69
CDK1 P06493 12/20 0.69
CCNB1 P14635 12/20 0.69
CCNB3 Q8WWL7 12/20 0.69
MAPT P10636 5/20 0.64
LMNA P02545 3/20 0.64
TDP1 Q9NUW8 2/20 0.64
HTT P42858 1/20 0.64
NCOA1 Q15788 1/20 0.64
NCOA3 Q9Y6Q9 1/20 0.64
SRC P12931 2/20 0.49
FLT4 P35916 2/20 0.49
MAPK1 P28482 2/20 0.49
CDC7 O00311 1/20 0.49
PLK4 O00444 1/20 0.49
IKBKB O14920 1/20 0.49
PDPK1 O15530 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688422 0.81 GSK3B (1.00) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL30319858 0.81 GSK3B (1.00) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL6239759 0.78 MAPT (1.00) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL4552964 0.76 CDK1 (0.62) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL20920125 0.72 GABRA1 (0.59) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL5263677 0.70 MAPT (0.69) GSK3BCDK5CCNB2CDK1CCNB1
SCHEMBL29855719 0.70 MAPT (0.69) GSK3BCDK5CCNB2CDK1CCNB1
SCHEMBL4162219 0.70 MAPT (0.69) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL21828647 0.69 CTSV (0.70) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL16301433 0.67 HTR2A (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999065910-A9 FUSED AZEPINONE CYCLIN DEPENDENT KINASE INHIBITORS US HEALTH (US) 2000-03-16 WO claimed