SCHEMBL7399245

SCHEMBL7399245

Oc1cc(C(F)(F)F)nn1-c1ccc2ccccc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.42
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PTGS1 P23219 1/20 0.39
PDPK1 O15530 6/20 0.38
PDE10A Q9Y233 3/20 0.38
ALDH1A1 P00352 3/20 0.37
HTR3E A5X5Y0 2/20 0.37
KDM4E B2RXH2 2/20 0.37
HTR3B O95264 2/20 0.37
CYP1A2 P05177 2/20 0.37
HTR3A P46098 2/20 0.37
HTR3D Q70Z44 2/20 0.37
HTR3C Q8WXA8 2/20 0.37
USP2 O75604 1/20 0.37
ADRB1 P08588 1/20 0.37
CYP3A4 P08684 1/20 0.37
HTR1A P08908 1/20 0.37
HTR2C P28335 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7405167 0.79 IRAK4 (0.42) PTGS1ALDH1A1KDM4EMAPTKMT2A
SCHEMBL537351 0.78 PDPK1 (0.50) RAB9APTGS1PDPK1ALDH1A1CYP1A2
SCHEMBL537395 0.75 PTGS1 (0.65) PTGS1PDPK1ALDH1A1KDM4ECYP1A2
SCHEMBL537523 0.75 TGFBR1 (0.44) RAB9APTGS1ALDH1A1KDM4EMAPK1
SCHEMBL7330567 0.73 PTGS1 (0.63) PTGS1PDPK1ALDH1A1KDM4ECYP1A2
SCHEMBL537761 0.72 MAPK1 (0.50) NPC1RAB9APTGS1ALDH1A1MAPK1
SCHEMBL31199040 0.71 CRACR2A (0.42) CNR2
SCHEMBL31199062 0.71 MAPT (0.44) CNR2NPC1RAB9AALDH1A1KDM4E
SCHEMBL7407050 0.71 PTGS1 (0.39) RAB9APTGS1ALDH1A1CYP1A2CYP3A4
SCHEMBL7405141 0.70 PTGS1 (0.44) CNR2PTGS1PDPK1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750550-A RESPIRATORY SYSTEM DISORDERS SANOFI (FR) 1998-05-12 US disclosed
WO-1997010243-A1 2-(PYRAZOL-5-YL-OXYMETHYL)-1,2-BENZISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SANOFI (US) 1997-03-20 WO disclosed