SCHEMBL7399397

SCHEMBL7399397

CC(CCC(=O)NCC#N)Cc1csc(-c2ccc(N3CCNCC3)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSL P07711 12/20 0.49
CTSS P25774 11/20 0.49
CTSB P07858 11/20 0.49
CTSK P43235 11/20 0.49
MAPKAPK2 P49137 1/20 0.44
AOC3 Q16853 1/20 0.37
CHEK1 O14757 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7394745 0.80 CTSL (0.59) CTSLCTSSCTSBCTSK
SCHEMBL4711786 0.76 CTSK (0.69) CTSLCTSSCTSBCTSK
SCHEMBL7397511 0.76 CTSL (0.51) CTSLCTSSCTSBCTSK
SCHEMBL7446518 0.76 CTSL (0.64) CTSLCTSSCTSBCTSK
SCHEMBL7436831 0.74 CTSL (0.64) CTSLCTSSCTSBCTSK
SCHEMBL7405812 0.70 CTSK (0.62) CTSLCTSSCTSBCTSKAOC3
SCHEMBL4701852 0.68 CTSK (0.69) CTSLCTSSCTSBCTSK
SCHEMBL7442354 0.67 CTSL (0.48) CTSLCTSSCTSBCTSK
SCHEMBL7439946 0.67 CTSK (0.51) CTSLCTSSCTSBCTSKAOC3
SCHEMBL7404362 0.66 CTSK (0.50) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001049288-A9 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2001-10-25 WO claimed