SCHEMBL7404362

SCHEMBL7404362

CC(CCC(=O)NCC#N)Cc1cccc(N2CCN(C)CC2)c1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.50
CTSL P07711 5/20 0.50
CTSB P07858 7/20 0.47
CTSS P25774 7/20 0.46
PRKD1 Q15139 2/20 0.43
AGXT P21549 1/20 0.42
MAPK14 Q16539 1/20 0.40
PLOD2 O00469 1/20 0.40
PLOD3 O60568 1/20 0.40
PLOD1 Q02809 1/20 0.40
HTR2C P28335 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447450 0.96 CTSK (0.54) CTSKCTSLCTSBCTSSPRKD1
SCHEMBL7405812 0.89 CTSK (0.62) CTSKCTSLCTSBCTSSPRKD1
SCHEMBL7442354 0.89 CTSL (0.48) CTSKCTSLCTSBCTSSAGXT
SCHEMBL7397511 0.85 CTSL (0.51) CTSKCTSLCTSBCTSS
SCHEMBL7439946 0.85 CTSK (0.51) CTSKCTSLCTSBCTSS
SCHEMBL7401645 0.81 CTSL (0.60) CTSKCTSLCTSBCTSSPRKD1
SCHEMBL7398927 0.79 CTSK (0.63) CTSKCTSLCTSBCTSSPRKD1
SCHEMBL7394745 0.79 CTSL (0.59) CTSKCTSLCTSBCTSS
SCHEMBL7451409 0.76 CTSB (0.53) CTSKCTSLCTSBCTSSPRKD1
SCHEMBL7444865 0.76 CTSK (0.39) CTSKCTSLCTSBCTSSPRKD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001049288-A9 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2001-10-25 WO claimed
WO-2001049288-A9 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2001-10-25 WO disclosed