Iodide

Iodide

SCHEMBL7399488

CSC1=Nc2ccccc2Cc2ccsc21.I

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 known ✓ P11229 1/20 0.30
CHRM3 known ✓ P20309 1/20 0.30
HRH4 Q9H3N8 2/20 0.38
DRD1 P21728 3/20 0.34
DRD3 P35462 3/20 0.34
DRD2 P14416 2/20 0.34
DRD4 P21917 2/20 0.34
DRD5 P21918 2/20 0.34
TRPA1 O75762 1/20 0.33
NOS3 P29474 2/20 0.31
NOS2 P35228 2/20 0.31
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM4 P08173 1/20 0.30
CYP3A4 P08684 1/20 0.30
CHRM5 P08912 1/20 0.30
ADRA2A P08913 1/20 0.30
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11872463 0.75 HRH4 (0.38) HRH4DRD1DRD3DRD2DRD4
SCHEMBL7420397 0.75 NOS2 (0.49) HRH4DRD1DRD3DRD2DRD4
Iodide SCHEMBL7585154 0.72 BACE1 (0.34) DRD1DRD3DRD2TRPA1LMNA
SCHEMBL11855700 0.71 HRH4 (0.66) HRH4DRD1DRD3DRD2DRD4
SCHEMBL11877889 0.67 HRH4 (0.49) HRH4DRD1DRD3DRD2DRD4
SCHEMBL10026452 0.67 HRH4 (0.40) HRH4TRPA1NOS3NOS2LMNA
SCHEMBL9409761 0.65 HRH1 (0.47) HRH4DRD1DRD3DRD2DRD4
SCHEMBL30310960 0.65 HRH1 (0.47) HRH4DRD1DRD3DRD2DRD4
SCHEMBL11861754 0.65 TRPA1 (0.55) HRH4DRD1DRD3DRD2DRD4
SCHEMBL3290813 0.64 MAOA (0.46) HRH4DRD1DRD3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000073313-A1 NEW TRICYCLIC AMIDINE DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2000-12-07 WO disclosed
WO-2000073312-A1 COMPOUNDS ASTRAZENECA AB (SE) 2000-12-07 WO disclosed