SCHEMBL7399753

SCHEMBL7399753

CC(C)C(=O)Nc1ccc(-c2c[nH]c(=O)cn2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.46
NPC1 O15118 6/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
KDM4E B2RXH2 4/20 0.45
POLB P06746 2/20 0.45
MAPT P10636 2/20 0.45
PTPN1 P18031 1/20 0.45
ALDH1A1 P00352 6/20 0.44
GAA P10253 1/20 0.44
RXFP1 Q9HBX9 1/20 0.43
HPGD P15428 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TP53 P04637 1/20 0.42
GLA P06280 1/20 0.42
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2778375 0.85 XDH (0.52) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL7397793 0.82 ALDH1A1 (0.44) KMT2APOLBPTPN1ALDH1A1
SCHEMBL7398696 0.82 DYRK1B (0.47) NPC1MAPTPTPN1ALDH1A1GAA
SCHEMBL7368321 0.81 NPC1 (0.50) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL7365549 0.81 TSHR (0.45) KDM4EPTPN1CA12CA1CA2
SCHEMBL7403582 0.81 RAB9A (0.47) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL7396486 0.80 ROCK2 (0.58) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL7366309 0.79 NPC1 (0.48) RAB9ANPC1SMN1; SMN2KMT2AMEN1
SCHEMBL7399852 0.79 KIT (0.46)
SCHEMBL7403608 0.78 PDE3B (0.48) RAB9ANPC1SMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0096517-A2 Aryl pyrazinones SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1983-12-21 EP claimed
US-4657906-A CARDIOVASCULAR DISORDERS SMITH KLINE & FRENCH LABORATORIES LTD. (GB) 1987-04-14 US disclosed
US-4556711-A CARDIOTONIC AGENTS SMITH KLINE & FRENCH LABORATORIES LTD. (US) 1985-12-03 US disclosed
EP-0096517-A2 Aryl pyrazinones SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1983-12-21 EP disclosed