Clofentezine

Clofentezine

SCHEMBL74002

Clc1ccccc1-c1nnc(-c2ccccc2Cl)nn1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.59
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
HPGD P15428 3/20 0.56
TP53 P04637 3/20 0.56
CYP2A6 P11509 1/20 0.52
ALDH1A1 P00352 3/20 0.52
HSD11B1 P28845 3/20 0.52
LMNA P02545 2/20 0.52
NOTUM Q6P988 1/20 0.48
TSHR P16473 2/20 0.47
HSD17B10 Q99714 3/20 0.47
KDM4E B2RXH2 2/20 0.47
IDO1 P14902 1/20 0.45
HSP90AA1 P07900 1/20 0.44
NFKB1 P19838 1/20 0.44
CASP3 P42574 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clofentezine SCHEMBL5022593 1.00 LDHA (0.59) LDHANPC1RAB9ASMN1; SMN2HPGD
Clofentezine SCHEMBL30917908 1.00 LDHA (0.59) LDHANPC1RAB9ASMN1; SMN2HPGD
Clofentezine SCHEMBL29375770 1.00 LDHA (0.59) LDHANPC1RAB9ASMN1; SMN2HPGD
Clofentezine SCHEMBL28407354 0.97 LDHA (0.57) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL9232863 0.89 LDHA (0.50) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL11255465 0.89 RAB9A (0.61) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL11405650 0.87 LDHA (0.48) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL22357676 0.87 HSD11B1 (0.52) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL11411501 0.87 CYP2A6 (0.64) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL18920574 0.87 LDHA (0.48) LDHANPC1RAB9ASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 17318 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4719059-A1 INCREASED PALATABILITY OF INSECTICIDAL INSECT BAITS Bio Logic Crop Science, S.L. (ES) 2026-04-08 EP claimed
US-20260083129-A1 PYRAZOLE AMIDE INSECTICIDES FMC CORP (US) 2026-03-26 US claimed
EP-4710766-A1 MIXTURES OF AMBRUTICIN WITH AT LEAST ONE FURTHER PESTICIDE BASF SE (DE) 2026-03-18 EP claimed
EP-4697936-A1 METHOD FOR THE PRODUCTION OF DIETARY FIBERS INTENDED FOR THE FOOD INDUSTRY Industrie Rolli Alimentari S.p.A. (IT) 2026-02-25 EP claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
US-20250351818-A1 PESTICIDAL BAIT COMPOSITION AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE, LLC (US) 2025-11-20 US claimed
US-12471599-B2 Agricultural compositions comprising remodeled nitrogen fixing microbes PIVOT BIO, INC. (US) 2025-11-18 US claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
US-20250338849-A1 FUNGICIDAL MIXTURE COMPRISING SUBSTITUTED PYRIDINES BASF SE (DE) 2025-11-06 US claimed
WO-2025223904-A1 MIXTURES OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS WITH AT LEAST ONE FURTHER PESTICIDE I BASF SE (DE) 2025-10-30 WO claimed
EP-0412937-A1 Plant acaricide CIBA-GEIGY AG (CH) 1991-02-13 EP claimed
EP-0381691-A1 LATEX-BASED AGRICULTURAL COMPOSITIONS. DOW CHEMICAL CO (GB) 1990-08-16 EP claimed
US-4912099-A Mixture of clofentezine and fenbutatin SCHERING AGROCHEMICALS LIMITED (GB) 1990-03-27 US claimed
WO-1989003176-A1 LATEX-BASED AGRICULTURAL COMPOSITIONS DOW CHEMICAL COMPANY LIMITED (GB) 1989-04-20 WO claimed
CN-88103536-A Miticide 1988-12-28 CN claimed
EP-0295790-A2 Acaricide formulations SCHERING AGROCHEMICALS LIMITED (GB) 1988-12-21 EP claimed
EP-0242502-A2 Pesticidal compositions HOECHST AKTIENGESELLSCHAFT (DE) 1987-10-28 EP claimed
EP-0005912-B1 ACARICIDAL, LARVICIDAL AND OVICIDAL TETRAZINE DERIVATIVES AND COMPOSITIONS, PROCESSES FOR THEIR PREPARATION AND METHODS OF USING THEM FBC LIMITED (GB) 1982-07-14 EP claimed
US-4237127-A MITICIDES, LARVICIDES, OVICIDES FISONS LIMITED (GB) 1980-12-02 US claimed
EP-0005912-A1 Acaricidal, larvicidal and ovicidal tetrazine derivatives and compositions, processes for their preparation and methods of using them FBC LIMITED (GB) 1979-12-12 EP claimed