Clofentezine

Clofentezine

SCHEMBL29375770

Clc1ccccc1-c1nnc(-c2ccccc2Cl)nn1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.59
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
HPGD P15428 3/20 0.56
TP53 P04637 3/20 0.56
CYP2A6 P11509 1/20 0.52
ALDH1A1 P00352 3/20 0.52
HSD11B1 P28845 3/20 0.52
LMNA P02545 2/20 0.52
NOTUM Q6P988 1/20 0.48
TSHR P16473 2/20 0.47
HSD17B10 Q99714 3/20 0.47
KDM4E B2RXH2 2/20 0.47
IDO1 P14902 1/20 0.45
HSP90AA1 P07900 1/20 0.44
NFKB1 P19838 1/20 0.44
CASP3 P42574 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clofentezine SCHEMBL5022593 1.00 LDHA (0.59) LDHANPC1RAB9ASMN1; SMN2HPGD
Clofentezine SCHEMBL30917908 1.00 LDHA (0.59) LDHANPC1RAB9ASMN1; SMN2HPGD
Clofentezine SCHEMBL74002 1.00 LDHA (0.59) LDHANPC1RAB9ASMN1; SMN2HPGD
Clofentezine SCHEMBL28407354 0.97 LDHA (0.57) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL9232863 0.89 LDHA (0.50) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL11255465 0.89 RAB9A (0.61) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL11405650 0.87 LDHA (0.48) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL22357676 0.87 HSD11B1 (0.52) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL11411501 0.87 CYP2A6 (0.64) LDHANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL18920574 0.87 LDHA (0.48) LDHANPC1RAB9ASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 377 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4734762-A1 BAIT COMPOSITIONS FMC Corporation (US) 2026-05-06 EP claimed
US-20260083130-A1 NOVEL SULFONATE BENZAMIDE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS FMC CORP (US) 2026-03-26 US claimed
US-12568969-B2 Pyridine compounds for controlling invertebrate pests FMC CORPORATION (US) 2026-03-10 US claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
US-12471599-B2 Agricultural compositions comprising remodeled nitrogen fixing microbes PIVOT BIO, INC. (US) 2025-11-18 US claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-4638432-A1 AZOLE COMPOUNDS FOR CONTROLLING AND COMBATING INVERTEBRATE PESTS FMC Corporation (US) 2025-10-29 EP claimed
EP-4640053-A2 MIXTURES COMPRISING INDAZOLE PESTICIDES FMC Corporation (US) 2025-10-29 EP claimed
US-20250287942-A1 FORMULATIONS FOR REPELLING BEES AND OTHER INSECTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-09-18 US claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
WO-2022164857-A1 AZOLE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS FMC CORPORATION (US) 2022-08-04 WO claimed
EP-4031530-A1 META-DIAMIDE INSECTICIDES FMC CORPORATION (US) 2022-07-27 EP claimed
EP-4013223-A1 MATERIAL DELIVERY SYSTEMS AND METHODS FMC Corporation (US) 2022-06-22 EP claimed
US-11339154-B2 Heterocycle-substituted bicyclic azole pesticides FMC CORPORATION (US) 2022-05-24 US claimed
EP-3996508-A1 MIXTURES COMPRISING INDAZOLE PESTICIDES FMC Corporation (US) 2022-05-18 EP claimed
US-20220135562-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES FMC CORPORATION 2022-05-05 US claimed
EP-3424919-B1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES FMC CORP (US) 2022-04-27 EP claimed
EP-3567036-B1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES FMC CORP (US) 2022-04-13 EP claimed
EP-3621964-B1 MESOIONIC INSECTICIDES FMC CORP (US) 2022-03-02 EP claimed
US-20220041582-A1 ISOXAZOLINE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS FMC CORPORATION 2022-02-10 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250287942-A1 FORMULATIONS FOR REPELLING BEES AND OTHER INSECTS ACHE, BCHE, DDT LDHA 3997/4885NPC1 505/4885RAB9A 2782/4885
US-20220041582-A1 ISOXAZOLINE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS PRDX1, CYP4X1, ACHE LDHA 4432/4885NPC1 2675/4885RAB9A 549/4885
US-11339154-B2 Heterocycle-substituted bicyclic azole pesticides DDT, NOX3, CYP4X1 LDHA 4487/4885NPC1 4115/4885RAB9A 2251/4885
US-12568969-B2 Pyridine compounds for controlling invertebrate pests COX6C, CCR1, CBR3 LDHA 4622/4885NPC1 1224/4885RAB9A 340/4885
US-12471599-B2 Agricultural compositions comprising remodeled nitrogen fixing microbes MYB, NANS, NANP LDHA 2548/4885NPC1 3966/4885RAB9A 2263/4885
US-20220135562-A1 HETEROCYCLE-SUBSTITUTED BICYCLIC AZOLE PESTICIDES DDT, NOX3, CYP4X1 LDHA 4487/4885NPC1 4115/4885RAB9A 2251/4885
US-20260083130-A1 NOVEL SULFONATE BENZAMIDE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS CBR1, CBR3, COX6B1 LDHA 3996/4885NPC1 1769/4885RAB9A 565/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.