SCHEMBL7400459

SCHEMBL7400459

O=C(Nc1cccc(Oc2ccccc2)c1)C(CCc1ccccc1)NC(=O)C1(C(=O)O)CCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.44
MMP3 P08254 1/20 0.44
MMP10 P09238 1/20 0.44
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
MMP12 P39900 1/20 0.44
MMP13 P45452 1/20 0.44
MMP14 P50281 1/20 0.44
S1PR1 P21453 2/20 0.44
MITF O75030 1/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
HPGD P15428 2/20 0.43
FFAR1 O14842 4/20 0.43
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400552 0.91 MAPT (0.42) MMP2MMP3MMP10MMP9MMP8
SCHEMBL7405755 0.87 HDAC8 (0.42) MMP2MMP3MMP10MMP9MMP8
SCHEMBL7402816 0.82 CASP3 (0.48)
SCHEMBL7408787 0.80 HDAC8 (0.58)
SCHEMBL7402346 0.79 HDAC1 (0.44) MMP2MMP3MMP10MMP9MMP8
SCHEMBL7406759 0.78 MMP2 (0.41) MMP2MMP3MMP10MMP9MMP8
SCHEMBL7408486 0.78 CASP3 (0.45) MMP2MMP3MMP10MMP9MMP8
SCHEMBL7402840 0.78 CASP3 (0.41)
SCHEMBL7409945 0.78 F10 (0.41) ALDH1A1HPGD
SCHEMBL7410069 0.77 HDAC4 (0.33) MMP2MMP3MMP10MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed