SCHEMBL7400552

SCHEMBL7400552

CCOC(=O)C1(C(=O)NC(CCc2ccccc2)C(=O)Nc2cccc(Oc3ccccc3)c2)CCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.42
LMNA P02545 2/20 0.42
HPGD P15428 2/20 0.42
RAB9A P51151 2/20 0.42
S1PR2 O95136 1/20 0.41
FFAR1 O14842 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TP53 P04637 1/20 0.41
MMP2 P08253 1/20 0.41
MMP3 P08254 1/20 0.41
MMP10 P09238 1/20 0.41
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
MMP12 P39900 1/20 0.41
MMP13 P45452 1/20 0.41
MMP14 P50281 1/20 0.41
S1PR1 P21453 1/20 0.41
HDAC4 P56524 2/20 0.40
MEF2D Q14814 2/20 0.40
EP300 Q09472 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7400459 0.91 MMP2 (0.44) MAPTLMNAHPGDRAB9AS1PR2
SCHEMBL7410624 0.83 HDAC4 (0.41) MAPTLMNAHPGDRAB9AS1PR2
SCHEMBL7405755 0.81 HDAC8 (0.42) HPGDALDH1A1MMP2MMP3MMP10
SCHEMBL7409945 0.81 F10 (0.41) HPGDALDH1A1HDAC4KMT2AMEN1
SCHEMBL7402816 0.78 CASP3 (0.48)
SCHEMBL7408787 0.77 HDAC8 (0.58) HDAC4
SCHEMBL7402840 0.76 CASP3 (0.41)
SCHEMBL7408486 0.74 CASP3 (0.45) HPGDALDH1A1MMP2MMP3MMP10
SCHEMBL7406759 0.74 MMP2 (0.41) HPGDS1PR2ALDH1A1MMP2MMP3
SCHEMBL7410069 0.74 HDAC4 (0.33) LMNAS1PR2FFAR1MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed