SCHEMBL7405755

SCHEMBL7405755

O=C(CCC(NC(=O)C1(C(=O)O)CCC1)C(=O)Nc1cccc(Oc2ccccc2)c1)OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
SIRT2 Q8IXJ6 4/20 0.42
CCKBR P32239 2/20 0.42
F10 P00742 1/20 0.41
PRSS1 P07477 1/20 0.41
SIRT5 Q9NXA8 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7409945 0.90 F10 (0.41) HDAC8HDAC3HDAC4HDAC1HDAC7
SCHEMBL7400459 0.87 MMP2 (0.44) ALDH1A1HPGDS1PR1MMP2MMP3
SCHEMBL7411328 0.84 CASP3 (0.44)
SCHEMBL7402346 0.82 HDAC1 (0.44) HDAC8HDAC3HDAC4HDAC1HDAC7
SCHEMBL7400552 0.81 MAPT (0.42) HDAC4ALDH1A1HPGDMEN1KMT2A
SCHEMBL7451783 0.80 CASP3 (0.39) MMP8
SCHEMBL7408820 0.80 HDAC4 (0.53) HDAC8HDAC3HDAC4HDAC1HDAC7
SCHEMBL7404353 0.80 HDAC3 (0.55) HDAC8HDAC3HDAC4HDAC1HDAC7
SCHEMBL7405678 0.79 KDR (0.35) HDAC8HDAC3HDAC4HDAC1HDAC7
SCHEMBL7407960 0.78 LTA4H (0.56) HDAC8HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076968-A1 MALONATES AS INHIBITORS OF THE ICE/CED-6 FAMILY OF CYSTEINE PROTEASES NOVARTIS AG (CH) 2002-10-03 WO disclosed