SCHEMBL7400617

SCHEMBL7400617

Oc1c(F)cc(N2CCC3(C=Cc4ccccc4O3)CC2)cc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 12/20 0.49
HTR2B P41595 1/20 0.49
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
DRD2 P14416 1/20 0.42
HTR2A P28223 1/20 0.42
SCD O00767 1/20 0.41
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
AKR1B1 P15121 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7370885 0.76 HTR2C (0.62) HTR2CHTR2BADRA1DADRA1AADRA1B
SCHEMBL4275574 0.73 SCD (0.39) HTR2CHTR2BADRA1DADRA1AADRA1B
SCHEMBL3413391 0.73 HTR2C (0.62) HTR2CHTR2BADRA1DADRA1AADRA1B
SCHEMBL12481728 0.72 HTR2C (0.57) HTR2CHTR2BADRA1DADRA1AADRA1B
SCHEMBL3552550 0.70 HTR2C (0.72) HTR2CHTR2BADRA1DADRA1AADRA1B
SCHEMBL3709748 0.70 HTR2C (0.55) HTR2CHTR2BADRA1DADRA1AADRA1B
SCHEMBL8002464 0.70 ADRA1A (0.66) HTR2CHTR2BADRA1DADRA1AADRA1B
SCHEMBL1115308 0.69 HTR2C (0.70) HTR2CHTR2BADRA1DADRA1AADRA1B
SCHEMBL4275257 0.68 HDAC3 (0.58) HTR2CHTR2BADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL4269341 0.68 ADRA1D (0.54) HTR2CHTR2BADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1232160-A1 SPIRO(2H-1-BENZOPYRAN-2,4'-PIPERIDINE)DERIVATES AS GLYCINE TRANSPORT INHIBITORS Akzo Nobel N.V. (NL) 2002-08-21 EP disclosed
WO-2001036423-A1 SPIRO(2H-1-BENZOPYRAN-2,4'-PIPERIDINE) DERIVATES AS GLYCINE TRANSPORT INHIBITORS AKZO NOBEL N.V. (NL) 2001-05-25 WO disclosed