SCHEMBL7400643

SCHEMBL7400643

Cn1c(NCCC(CO)CO)nc2c1c(=O)n(CC1CC1)c(=O)n2CC1CC1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 12/20 0.55
PDE4A P27815 12/20 0.55
PDE4B Q07343 12/20 0.55
PDE4C Q08493 12/20 0.55
PDE4D Q08499 12/20 0.55
CYP2C19 P33261 1/20 0.43
TP53 P04637 2/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
ATM Q13315 1/20 0.39
KDM4E B2RXH2 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2D6 P10635 1/20 0.39
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7395398 0.86 PDE5A (0.49) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7400772 0.80 PDE5A (0.65) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7401994 0.74 PDE5A (0.42) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7400872 0.71 PDE5A (1.00) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7446384 0.69 PDE5A (1.00) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7399841 0.69 PDE5A (0.61) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7400585 0.67 PDE4A (1.00) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL25235156 0.65 PDE5A (0.60) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL25222680 0.64 PDE5A (0.59) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL24769075 0.64 LMNA (0.60) CYP2C19ALDH1A1LMNAHTTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641344-A1 8-SUBSTITUTED ANTHINES AS PHOSPHODIESTERASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1995-03-08 EP disclosed
WO-1993023401-A1 8-SUBSTITUTED ANTHINES AS PHOSPHODIESTERASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1993-11-25 WO disclosed