SCHEMBL7401210

SCHEMBL7401210

Nc1cccc(CC2=C(O)CC(CCc3ccccc3)(CCc3ccccc3)OC2=O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.42
MAOB P27338 2/20 0.42
SIGMAR1 Q99720 1/20 0.36
CYP19A1 P11511 1/20 0.35
GRM2 Q14416 1/20 0.35
GRM3 Q14832 1/20 0.35
MLNR O43193 1/20 0.35
NR1I2 O75469 1/20 0.35
ABCB11 O95342 1/20 0.35
PGR P06401 1/20 0.35
CTSD P07339 1/20 0.35
CHRM2 P08172 1/20 0.35
ADRA2A P08913 1/20 0.35
PGA5 P0DJD9 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CTSE P14091 1/20 0.35
GABRA1 P14867 1/20 0.35
ADRA2C P18825 1/20 0.35
DRD1 P21728 1/20 0.35
HTR2A P28223 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3632231 0.84 HTR2B (0.40) MAOAMAOBSIGMAR1CYP19A1MLNR
SCHEMBL8807657 0.84 HTR2B (0.40) MAOAMAOBSIGMAR1CYP19A1MLNR
SCHEMBL8805739 0.84 HTR2B (0.40) MAOAMAOBSIGMAR1CYP19A1MLNR
SCHEMBL8807004 0.83 MLNR (0.41) MAOAMAOBSIGMAR1CYP19A1GRM2
SCHEMBL7399940 0.82 SIGMAR1 (0.42) SIGMAR1AGTR1
SCHEMBL8808039 0.78 MLNR (0.34) MAOAMAOBCYP19A1MLNRNR1I2
SCHEMBL7402849 0.78 MLNR (0.56) MLNRNR1I2ABCB11PGRCTSD
SCHEMBL8805860 0.77 MAOA (0.35) MAOAMAOBSIGMAR1CYP19A1GRM2
SCHEMBL8809744 0.76 MLNR (0.38) CYP19A1MLNRNR1I2ABCB11PGR
SCHEMBL8809891 0.75 GRM2 (0.34) MAOAMAOBSIGMAR1CYP19A1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6169181-B1 HUMAN IMMUNODEFICIENCY VIRUS PROTEINASE INHIBITORS PHARMACIA & UPJOHN COMPANY 2001-01-02 US disclosed
US-5852195-A Pyranone compounds useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1998-12-22 US disclosed
EP-0758327-A1 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-19 EP disclosed
WO-1995030670-A2 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-16 WO disclosed