SCHEMBL8807657

SCHEMBL8807657

CCCC1(CCc2ccccc2)CC(O)=C(CCCc2cccc(N)c2)C(=O)O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.40
MLNR O43193 1/20 0.40
NR1I2 O75469 1/20 0.40
ABCB11 O95342 1/20 0.40
PGR P06401 1/20 0.40
CTSD P07339 1/20 0.40
CHRM2 P08172 1/20 0.40
ADRA2A P08913 1/20 0.40
PGA5 P0DJD9 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CTSE P14091 1/20 0.40
GABRA1 P14867 1/20 0.40
ADRA2C P18825 1/20 0.40
DRD1 P21728 1/20 0.40
HTR2A P28223 1/20 0.40
AGTR1 P30556 1/20 0.40
CCKAR P32238 1/20 0.40
ADRA1A P35348 1/20 0.40
PTGS2 P35354 1/20 0.40
PPARG P37231 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3632231 1.00 HTR2B (0.40) HTR2BMLNRNR1I2ABCB11PGR
SCHEMBL8805739 1.00 HTR2B (0.40) HTR2BMLNRNR1I2ABCB11PGR
SCHEMBL8805860 0.95 MAOA (0.35) HTR2BMLNRNR1I2ABCB11PGR
SCHEMBL9199813 0.91 MLNR (0.41) HTR2BMLNRNR1I2ABCB11PGR
SCHEMBL8807004 0.87 MLNR (0.41) HTR2BMLNRNR1I2ABCB11PGR
SCHEMBL8807543 0.85 MLNR (0.43) HTR2BMLNRNR1I2ABCB11PGR
SCHEMBL8806724 0.85 OPRD1 (0.40) HTR2BMLNRNR1I2ABCB11PGR
SCHEMBL7401210 0.84 MAOA (0.42) HTR2BMLNRNR1I2ABCB11PGR
SCHEMBL8809891 0.82 GRM2 (0.34) MAOAMAOBSIGMAR1CYP19A1
SCHEMBL8808265 0.81 CRHBP (0.39) HTR2BMLNRNR1I2ABCB11PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758327-A1 PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1997-02-19 EP disclosed