SCHEMBL7401341

SCHEMBL7401341

O=CNc1ccc(Br)cc1Oc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.66
ADORA3 P0DMS8 2/20 0.44
PTGS1 P23219 2/20 0.44
MIF P14174 1/20 0.44
PDE4A P27815 1/20 0.44
PDE4D Q08499 1/20 0.44
SLC6A4 P31645 2/20 0.43
HTR6 P50406 1/20 0.43
LMNA P02545 4/20 0.41
KMT2A Q03164 4/20 0.41
GAA P10253 1/20 0.41
HTT P42858 2/20 0.40
MEN1 O00255 3/20 0.39
TTR P02766 1/20 0.38
MAPT P10636 3/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2C9 P11712 2/20 0.37
MAPK1 P28482 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3521281 0.88 TSHR (0.66) TSHRADORA3PTGS1MIFPDE4A
SCHEMBL4414857 0.80 TSHR (1.00) TSHRADORA3PTGS1MIFPDE4A
SCHEMBL12946520 0.77 HTT (0.50) TSHRLMNAKMT2AGAAHTT
SCHEMBL29182671 0.76 ALDH1A1 (0.52) TSHRLMNAKMT2AGAAMEN1
SCHEMBL4464378 0.76 LMNA (0.62) TSHRSLC6A4HTR6LMNAKMT2A
SCHEMBL28402042 0.74 TRIM24 (0.52) TSHRADORA3PTGS1SLC6A4LMNA
SCHEMBL20561801 0.73 HPGD (0.44) TSHRLMNAKMT2AGAAHTT
SCHEMBL2075254 0.72 LMNA (0.62) TSHRSLC6A4HTR6LMNAKMT2A
SCHEMBL811731 0.72 SLC6A4 (0.53) TSHRSLC6A4HTR6LMNAKMT2A
SCHEMBL1128732 0.72 TSHR (0.66) TSHRLMNAKMT2AHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6008213-A A INHIBITOR OF VITRONECTIN RECEPTOR AND FIBRINOGEN RECEPTOR; USEFUL FOR INHIBITING PLATELET AGGREGATION AND OSTEOPOROSIS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-28 US disclosed
EP-0910563-A1 INTEGRIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-04-28 EP disclosed
EP-0910563-A4 1999-04-28 EP disclosed
WO-1997001540-A1 INTEGRIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-01-16 WO disclosed