SCHEMBL7401359

SCHEMBL7401359

Cc1cc(CCOc2ccc(C(=O)N3CCCC(C(=O)NO)C3)cc2)c2ccccc2n1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 3/20 0.61
MMP2 P08253 3/20 0.51
MMP9 P14780 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6595607 0.92 ADAM17 (0.72) ADAM17MMP2
SCHEMBL7399667 0.89 ADAM17 (0.60) ADAM17MMP2MMP9
SCHEMBL6594904 0.83 ADAM17 (0.60) ADAM17MMP2
SCHEMBL6597332 0.83 MMP2 (0.65) ADAM17MMP2MMP9
SCHEMBL7401362 0.82 ADAM17 (0.51) ADAM17MMP2MMP9
SCHEMBL6598735 0.80 ADAM17 (0.70) ADAM17MMP2MMP9
SCHEMBL7403330 0.77 ADAM17 (0.54) ADAM17MMP2MMP9
SCHEMBL7535624 0.76 MMP2 (0.76) ADAM17MMP2MMP9
SCHEMBL7535633 0.76 MMP2 (0.76) ADAM17MMP2MMP9
SCHEMBL7535643 0.76 MMP2 (0.76) ADAM17MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263756-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA Bristol-Myers Squibb Pharma Company (US) 2002-12-11 EP disclosed
WO-2001070734-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-09-27 WO disclosed