SCHEMBL7401362

SCHEMBL7401362

Cc1cc(C(C)Oc2ccc(C(=O)N3CCCC(C(=O)NO)C3)cc2)c2ccccc2n1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 2/20 0.51
LMNA P02545 2/20 0.47
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPK1 P28482 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HPGD P15428 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MMP2 P08253 2/20 0.43
MMP9 P14780 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399671 0.88 ADAM17 (0.51) ADAM17LMNAKDM4ENPC1ALDH1A1
SCHEMBL6595607 0.83 ADAM17 (0.72) ADAM17MMP2
SCHEMBL7401359 0.82 ADAM17 (0.61) ADAM17MMP2MMP9
SCHEMBL7535614 0.76 MMP2 (0.64) ADAM17MMP2MMP9
SCHEMBL6629887 0.75 SMN1; SMN2 (0.49) KDM4ENPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL6594904 0.74 ADAM17 (0.60) ADAM17MMP2
SCHEMBL6597332 0.74 MMP2 (0.65) ADAM17MMP2MMP9
SCHEMBL7430037 0.73 ADAM17 (0.75) ADAM17MMP2MMP9
SCHEMBL6633286 0.73 SMN1; SMN2 (0.47) KDM4ENPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL6598735 0.72 ADAM17 (0.70) ADAM17MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1263756-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA Bristol-Myers Squibb Pharma Company (US) 2002-12-11 EP disclosed
WO-2001070734-A2 BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-09-27 WO disclosed