SCHEMBL7401360

SCHEMBL7401360

COC(=O)C(Cc1ccc2c(c1)OCO2)=C(c1ccc(OC)cc1)c1ccc(OC)cc1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.60
RAB9A P51151 4/20 0.57
NPC1 O15118 3/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
LMNA P02545 1/20 0.56
HPGD P15428 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
EDNRB P24530 4/20 0.55
EDNRA P25101 3/20 0.53
MAPT P10636 1/20 0.52
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7404248 0.89 EDNRB (0.61) ALDH1A1RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL7397215 0.88 ALDH1A1 (0.52) ALDH1A1RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL25203201 0.83 RAB9A (0.70) ALDH1A1RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL7401629 0.81 HPGD (0.51) ALDH1A1RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL14518414 0.80 ALDH1A1 (0.70) ALDH1A1RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL8736580 0.77 ALDH1A1 (0.68) ALDH1A1RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL7399206 0.76 ALDH1A1 (0.66) ALDH1A1RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL27981072 0.75 RAB9A (0.87) ALDH1A1RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL389405 0.75 SMN1; SMN2 (0.66) ALDH1A1RAB9ANPC1SMN1; SMN2LMNA
SCHEMBL26624014 0.75 KMT2A (0.72) ALDH1A1RAB9ANPC1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0650484-B1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2000-01-26 EP disclosed
US-5559105-A ANTAGONIST FOR ENDOTHELIN RECEPTORS, HYPOTENSIVE AGENTS, TREATMENT OF KIDNEY FAILURE OR CEREBROVASCULAR DISORDERS SMITHKLINE BEECHAM CORPORATION (US) 1996-09-24 US disclosed
EP-0650484-A1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1995-05-03 EP disclosed
WO-1994002474-A1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-02-03 WO disclosed