SCHEMBL7401645

SCHEMBL7401645

CC(CCC(=O)NCC#N)Cc1cccc(-c2csc(N3CCN(C)CC3)n2)c1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSL P07711 7/20 0.60
CTSK P43235 7/20 0.60
CTSB P07858 6/20 0.60
CTSS P25774 6/20 0.60
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 6/20 0.44
LMNA P02545 4/20 0.44
ALDH1A1 P00352 4/20 0.44
PRKD1 Q15139 1/20 0.44
KDM4E B2RXH2 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MAPK1 P28482 3/20 0.42
HTT P42858 2/20 0.41
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7398927 0.98 CTSK (0.63) CTSLCTSKCTSBCTSSMEN1
SCHEMBL7436831 0.90 CTSL (0.64) CTSLCTSKCTSBCTSSMEN1
SCHEMBL7446518 0.87 CTSL (0.64) CTSLCTSKCTSBCTSSMAPT
SCHEMBL7392893 0.85 CTSL (0.55) CTSLCTSKCTSBCTSSMEN1
SCHEMBL7447450 0.83 CTSK (0.54) CTSLCTSKCTSBCTSSPRKD1
SCHEMBL7399341 0.82 CTSL (0.50) CTSLCTSKCTSBCTSSMEN1
SCHEMBL7405812 0.82 CTSK (0.62) CTSLCTSKCTSBCTSSPRKD1
SCHEMBL7404362 0.81 CTSK (0.50) CTSLCTSKCTSBCTSSPRKD1
SCHEMBL4718661 0.77 CTSK (0.97) CTSLCTSKCTSBCTSS
SCHEMBL4712046 0.75 CTSK (1.00) CTSLCTSKCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001049288-A9 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS MERCK FROSST CANADA INC (CA) 2001-10-25 WO claimed