SCHEMBL740294

SCHEMBL740294

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)Cc3ccc(-c4ccc5c(c4)NC(=O)C5)cc3)C2)nc2c(F)cccc21

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CFD P00746 3/20 0.37
SMYD3 Q9H7B4 1/20 0.34
PADI4 Q9UM07 2/20 0.33
DPP4 P27487 4/20 0.33
CPT1A P50416 2/20 0.32
CPT2 P23786 1/20 0.32
CYP2D6 P10635 1/20 0.32
HRH1 P35367 1/20 0.32
CRBN Q96SW2 1/20 0.32
MCHR1 Q99705 1/20 0.32
CTSC P53634 5/20 0.32
CTSK P43235 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL742026 1.00 CFD (0.37) CFDSMYD3PADI4DPP4CPT1A
SCHEMBL741416 0.95 CFD (0.36) CFDSMYD3PADI4CPT1ACPT2
SCHEMBL741417 0.95 CFD (0.36) CFDSMYD3PADI4CPT1ACPT2
SCHEMBL742244 0.90 CFD (0.34) CFDDPP4CYP2D6HRH1CTSC
SCHEMBL742245 0.90 CFD (0.34) CFDDPP4CYP2D6HRH1CTSC
SCHEMBL741798 0.89 LIPG (0.35) CFDPADI4CTSC
SCHEMBL741797 0.89 LIPG (0.35) CFDPADI4CTSC
SCHEMBL741966 0.88 AKT1 (0.36) CFDSMYD3PADI4CPT1ACPT2
SCHEMBL742052 0.88 AKT1 (0.36) CFDSMYD3PADI4CPT1ACPT2
SCHEMBL740771 0.88 HTT (0.39) CFDDPP4CYP2D6HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed