SCHEMBL740323

SCHEMBL740323

COCCCn1c(C2CCCN(C(=O)O)C2)nc2cccc(Cl)c21

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 10/20 0.42
HRH1 P35367 6/20 0.42
CYP2D6 P10635 5/20 0.42
CHRM1 P11229 3/20 0.41
TP53 P04637 1/20 0.38
HSD11B1 P28845 4/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
USP2 O75604 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740661 0.89 P2RX7 (0.41) TP53KMT2AMEN1
SCHEMBL740662 0.89 P2RX7 (0.41) TP53KMT2AMEN1
SCHEMBL739857 0.85 HRH1 (0.57) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL740437 0.83 HRH1 (0.38) KCNH2HRH1CYP2D6CHRM1HSD11B1
SCHEMBL740436 0.83 HRH1 (0.38) KCNH2HRH1CYP2D6CHRM1HSD11B1
SCHEMBL740778 0.82 MMEL1 (0.38) KCNH2HRH1CYP2D6CHRM1HSD11B1
SCHEMBL739361 0.82 HRH1 (0.35) KCNH2HRH1CYP2D6CHRM1HSD11B1
SCHEMBL739667 0.81 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1TP53
SCHEMBL739144 0.81 KCNH2 (0.38) KCNH2HRH1CYP2D6CHRM1ALDH1A1
SCHEMBL739145 0.81 KCNH2 (0.38) KCNH2HRH1CYP2D6CHRM1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed