SCHEMBL740324

SCHEMBL740324

COCCCn1c(C2CCCN(C(=O)OC(C)(C)C)C2)nc2ccncc21

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.44
KCNH2 Q12809 3/20 0.41
HRH1 P35367 2/20 0.41
CYP2D6 P10635 1/20 0.41
HPGDS O60760 2/20 0.41
NLRP3 Q96P20 2/20 0.40
GPR119 Q8TDV5 5/20 0.39
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
CHRM1 P11229 1/20 0.39
TRPV3 Q8NET8 1/20 0.38
SCN9A Q15858 1/20 0.38
USP30 Q70CQ3 1/20 0.37
CCNK O75909 1/20 0.37
CDK12 Q9NYV4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762625 1.00 CYP2C9 (0.44) CYP2C9KCNH2HRH1CYP2D6HPGDS
SCHEMBL741974 0.89 KCNH2 (0.52) KCNH2HRH1CYP2D6HPGDSCHRM1
SCHEMBL741975 0.89 KCNH2 (0.52) KCNH2HRH1CYP2D6HPGDSCHRM1
SCHEMBL741439 0.88 HRH1 (0.46) KCNH2HRH1CYP2D6NLRP3CHRM1
SCHEMBL741679 0.85 TRPV3 (0.41) KCNH2HRH1CYP2D6HPGDSCHRM1
SCHEMBL741680 0.85 TRPV3 (0.41) KCNH2HRH1CYP2D6HPGDSCHRM1
SCHEMBL762594 0.85 TRPV3 (0.43) KCNH2HRH1CYP2D6HPGDSALOX5AP
SCHEMBL742014 0.85 HTT (0.43) KCNH2HRH1CYP2D6CHRM1
SCHEMBL742013 0.85 HTT (0.43) KCNH2HRH1CYP2D6CHRM1
SCHEMBL765031 0.84 P2RX3 (0.45) KCNH2HRH1CYP2D6HPGDSCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed