SCHEMBL740397

SCHEMBL740397

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)Cc3ccc(-c4ccc5occc5c4)cc3)C2)nc2c(C)cccc21

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
TSHR P16473 3/20 0.36
KMT2A Q03164 1/20 0.36
GYS1 P13807 1/20 0.34
CTSC P53634 1/20 0.34
BTK Q06187 3/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
DYRK1A Q13627 1/20 0.34
FASN P49327 5/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
NPY1R P25929 1/20 0.32
CFD P00746 1/20 0.32
DPP4 P27487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740398 1.00 ALDH1A1 (0.36) ALDH1A1TSHRKMT2AGYS1CTSC
SCHEMBL739855 0.87 PIK3CD (0.37) CTSCBTKFASN
SCHEMBL739856 0.87 PIK3CD (0.37) CTSCBTKFASN
SCHEMBL738530 0.86 KMT2A (0.36) ALDH1A1TSHRKMT2ACTSCBTK
SCHEMBL740270 0.86 KMT2A (0.36) ALDH1A1TSHRKMT2ACTSCBTK
SCHEMBL738529 0.86 KMT2A (0.36) ALDH1A1TSHRKMT2ACTSCBTK
SCHEMBL739272 0.85 NPY1R (0.36) ALDH1A1TSHRKMT2ABTKNPY1R
SCHEMBL739273 0.85 NPY1R (0.36) ALDH1A1TSHRKMT2ABTKNPY1R
SCHEMBL741986 0.85 SMYD3 (0.35) ALDH1A1TSHRKMT2ACTSCBTK
SCHEMBL740638 0.85 GSK3B (0.37) BTKDYRK1ACFD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed