SCHEMBL741986

SCHEMBL741986

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)Cc3ccc(-c4ccc5c(c4)CC(=O)N5C)cc3)C2)nc2c(C)cccc21

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.35
CTSC P53634 3/20 0.35
PADI4 Q9UM07 2/20 0.34
BTK Q06187 2/20 0.33
CFD P00746 2/20 0.32
BMPR1A P36894 2/20 0.32
ACVRL1 P37023 2/20 0.32
ACVR1 Q04771 2/20 0.32
NPY1R P25929 3/20 0.32
BRD4 O60885 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
KMT2A Q03164 1/20 0.32
BMPR1B O00238 1/20 0.32
TGFBR1 P36897 1/20 0.32
KDM1A O60341 1/20 0.32
DPP4 P27487 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741987 1.00 SMYD3 (0.35) SMYD3CTSCPADI4BTKCFD
SCHEMBL742052 0.89 AKT1 (0.36) SMYD3PADI4BTKCFDNPY1R
SCHEMBL741966 0.89 AKT1 (0.36) SMYD3PADI4BTKCFDNPY1R
SCHEMBL738530 0.86 KMT2A (0.36) CTSCBTKCFDNPY1RALDH1A1
SCHEMBL738529 0.86 KMT2A (0.36) CTSCBTKCFDNPY1RALDH1A1
SCHEMBL740270 0.86 KMT2A (0.36) CTSCBTKCFDNPY1RALDH1A1
SCHEMBL740398 0.85 ALDH1A1 (0.36) CTSCBTKCFDNPY1RALDH1A1
SCHEMBL740397 0.85 ALDH1A1 (0.36) CTSCBTKCFDNPY1RALDH1A1
SCHEMBL741161 0.85 BTK (0.31) CTSCBTKCFDNPY1RBRD4
SCHEMBL741160 0.85 BTK (0.31) CTSCBTKCFDNPY1RBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed