SCHEMBL7405121

SCHEMBL7405121

CC(C)(C)OC(=O)NC1CCc2cc(OCC(=O)OCc3ccccc3)ccc2C1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.49
CA2 P00918 3/20 0.49
ACHE P22303 3/20 0.49
TAOK1 Q7L7X3 1/20 0.45
TAOK3 Q9H2K8 1/20 0.45
FAAH O00519 8/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RORC P51449 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
KLK7 P49862 1/20 0.42
KLK5 Q9Y337 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8767884 0.84 CA1 (0.55) CA1CA2ACHETAOK1TAOK3
SCHEMBL8767895 0.84 CA1 (0.55) CA1CA2ACHETAOK1TAOK3
SCHEMBL9443665 0.84 ADRB3 (0.51) CA1CA2ACHEALDH1A1POLB
SCHEMBL9443694 0.84 ADRB3 (0.51) CA1CA2ACHEALDH1A1POLB
SCHEMBL9443701 0.84 ADRB3 (0.51) CA1CA2ACHEALDH1A1POLB
SCHEMBL7406582 0.83 KDM4E (0.42) KMT2AALDH1A1KDM4ELMNAPOLB
SCHEMBL5679215 0.81 HDAC8 (0.53) CA1CA2ACHEKMT2AL3MBTL1
SCHEMBL7035289 0.81 MTNR1A (0.53) CA1CA2ACHE
SCHEMBL5681677 0.81 MTNR1A (0.53) CA1CA2ACHE
SCHEMBL8103696 0.79 FAAH (0.48) ACHEFAAHKDM4ELMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6117910-A Bicyclic fibrinogen antagonists SMITHKLINE BEECHAM CORPORATION (US) 2000-09-12 US disclosed
EP-0799189-A4 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-17 EP disclosed
EP-0799189-A1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-10-08 EP disclosed
WO-1996018602-A1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1996-06-20 WO disclosed