SCHEMBL7406451

SCHEMBL7406451

Cc1cc(NC(=O)c2ccc3cc(C=NN)ccc3c2)no1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 13/20 0.56
NPC1 O15118 11/20 0.56
SMN1; SMN2 Q16637 6/20 0.54
TP53 P04637 5/20 0.54
TSHR P16473 1/20 0.54
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
ALDH1A1 P00352 3/20 0.52
NPSR1 Q6W5P4 1/20 0.51
CYP1A2 P05177 1/20 0.50
CYP2C19 P33261 1/20 0.50
KDM4E B2RXH2 2/20 0.49
RXFP1 Q9HBX9 1/20 0.49
MAPK1 P28482 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7340325 0.81 GRM5 (0.56) RAB9ANPC1SMN1; SMN2TP53
SCHEMBL7334320 0.81 KDM4E (0.52) RAB9ANPC1SMN1; SMN2TP53TSHR
SCHEMBL7406442 0.79 NPC1 (0.63) RAB9ANPC1SMN1; SMN2TP53TSHR
SCHEMBL7336457 0.78 NPC1 (0.53) RAB9ANPC1SMN1; SMN2TP53TSHR
SCHEMBL7337895 0.78 DNM1 (0.38) RAB9ANPC1MEN1KMT2AKDM4E
SCHEMBL7346861 0.77 SIRT2 (0.53) RAB9ANPC1SMN1; SMN2TP53TSHR
SCHEMBL7341819 0.77 SIRT2 (0.54) RAB9ANPC1SMN1; SMN2TP53MEN1
SCHEMBL7334154 0.76 RAB9A (0.67) RAB9ANPC1SMN1; SMN2TP53MEN1
SCHEMBL7343154 0.76 MAPT (0.60) RAB9ANPC1SMN1; SMN2MEN1KMT2A
SCHEMBL7345841 0.75 ALDH1A1 (0.53) RAB9ANPC1SMN1; SMN2TP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20010049374-A1 Urokinase inhibitors STEELE ANDREW W (US) 2001-12-06 US disclosed
US-6284796-B1 NAPHTHAMIDINE COMPOUNDS ABBOTT LABORATORIES 2001-09-04 US disclosed
US-6258822-B1 ENZYME INHIBITORS OF NAPHTHALENE AMIDINE COMPOUNDS ABBOTT LABORATORIES 2001-07-10 US disclosed
EP-1000018-A2 UROKINASE INHIBITORS Abbott Laboratories (US) 2000-05-17 EP disclosed
WO-1999005096-A2 UROKINASE INHIBITORS ABBOTT LABORATORIES (US) 1999-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010049374-A1 Urokinase inhibitors SERPINE1, PLAU, SERPINB1 RAB9A 2845/4885NPC1 2478/4885SMN1; SMN2 1786/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.