SCHEMBL7407208

SCHEMBL7407208

NC(=S)c1ccc(C(=O)Nc2ccc(C(=O)O)cc2NC(=O)c2ccc3ccccc3c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
RAB9A P51151 3/20 0.53
TDP1 Q9NUW8 1/20 0.53
NR1H4 Q96RI1 4/20 0.53
KDM4E B2RXH2 1/20 0.51
PLAU P00749 2/20 0.50
DHODH Q02127 2/20 0.50
SLC16A3 O15427 1/20 0.50
F2 P00734 1/20 0.48
PLG P00747 1/20 0.48
PLAT P00750 1/20 0.48
KLKB1 P03952 1/20 0.48
KLK1 P06870 1/20 0.48
PRSS1 P07477 1/20 0.48
PPARG P37231 1/20 0.47
DEGS1 O15121 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414642 1.00 NPC1 (0.55) NPC1MEN1KMT2ARAB9ATDP1
SCHEMBL7411350 0.88 GPR27 (0.51) NPC1MEN1KMT2ASLC16A3F2
SCHEMBL7411445 0.86 ALDH1A1 (0.54) NPC1MEN1KMT2ARAB9ANR1H4
SCHEMBL7411398 0.86 ALDH1A1 (0.54) NPC1MEN1KMT2ARAB9ANR1H4
SCHEMBL7460237 0.85 NR1H4 (0.47) NPC1MEN1KMT2ARAB9ATDP1
SCHEMBL7413497 0.84 SLC16A3 (0.52) KMT2ASLC16A3F2PRSS1
SCHEMBL7409765 0.83 NPC1 (0.46) NPC1RAB9ATDP1NR1H4KDM4E
SCHEMBL7413259 0.83 MEN1 (0.56) NPC1MEN1KMT2ARAB9ATDP1
SCHEMBL7409183 0.81 MEN1 (0.84) NPC1MEN1KMT2ARAB9AKDM4E
SCHEMBL7410644 0.81 MEN1 (0.84) NPC1MEN1KMT2ARAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999042439-A1 NOVEL THIOBENZAMIDES ROCHE DIAGNOSTICS GMBH (DE) 1999-08-26 WO claimed
WO-1999042439-A1 NOVEL THIOBENZAMIDES ROCHE DIAGNOSTICS GMBH (DE) 1999-08-26 WO disclosed
EP-0937711-A1 Thiobenzamides, process for their preparation and medicaments containing them Roche Diagnostics GmbH (DE) 1999-08-25 EP disclosed