SCHEMBL740730

SCHEMBL740730

COCCCn1c(C2CCCN(C(=O)O)C2)nc2ccc(F)cc21

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 9/20 0.44
CYP2D6 P10635 7/20 0.44
KCNH2 Q12809 7/20 0.43
CHRM1 P11229 3/20 0.43
BRD4 O60885 3/20 0.41
MAPT P10636 3/20 0.41
TP53 P04637 1/20 0.41
ADORA2A P29274 1/20 0.40
USP2 O75604 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739667 0.89 KCNH2 (0.43) HRH1CYP2D6KCNH2CHRM1BRD4
SCHEMBL739392 0.89 KCNH2 (0.45) HRH1CYP2D6KCNH2CHRM1BRD4
SCHEMBL762594 0.89 TRPV3 (0.43) HRH1CYP2D6KCNH2CHRM1BRD4
SCHEMBL739857 0.87 HRH1 (0.57) HRH1CYP2D6KCNH2CHRM1USP2
SCHEMBL740454 0.86 ADORA2A (0.51) HRH1CYP2D6KCNH2CHRM1BRD4
SCHEMBL740966 0.84 KCNH2 (0.44) HRH1CYP2D6KCNH2CHRM1ADORA2A
SCHEMBL741439 0.84 HRH1 (0.46) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL740716 0.81 CYP2D6 (0.41) HRH1CYP2D6KCNH2CHRM1MAPT
SCHEMBL740717 0.81 CYP2D6 (0.41) HRH1CYP2D6KCNH2CHRM1MAPT
SCHEMBL739990 0.81 HRH1 (0.44) HRH1CYP2D6KCNH2CHRM1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed