SCHEMBL740716

SCHEMBL740716

COCCCn1c(C2CCCN(C(=O)OC(C)(C)C)C2)nc2cc(F)ccc21

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.41
HRH1 P35367 7/20 0.41
TRPV3 Q8NET8 1/20 0.41
KCNH2 Q12809 5/20 0.41
CHRM1 P11229 2/20 0.41
ALOX5AP P20292 1/20 0.40
FEN1 P39748 1/20 0.40
HPGDS O60760 1/20 0.40
MAPT P10636 2/20 0.40
SCN9A Q15858 2/20 0.40
TP53 P04637 1/20 0.40
P2RX3 P56373 1/20 0.39
P2RX2 Q9UBL9 1/20 0.39
USP30 Q70CQ3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740717 1.00 CYP2D6 (0.41) CYP2D6HRH1TRPV3KCNH2CHRM1
SCHEMBL762594 0.93 TRPV3 (0.43) CYP2D6HRH1TRPV3KCNH2CHRM1
SCHEMBL765031 0.91 P2RX3 (0.45) CYP2D6HRH1TRPV3KCNH2CHRM1
SCHEMBL741975 0.88 KCNH2 (0.52) CYP2D6HRH1KCNH2CHRM1HPGDS
SCHEMBL741974 0.88 KCNH2 (0.52) CYP2D6HRH1KCNH2CHRM1HPGDS
SCHEMBL741680 0.85 TRPV3 (0.41) CYP2D6HRH1TRPV3KCNH2CHRM1
SCHEMBL742013 0.85 HTT (0.43) CYP2D6HRH1KCNH2CHRM1MAPT
SCHEMBL742014 0.85 HTT (0.43) CYP2D6HRH1KCNH2CHRM1MAPT
SCHEMBL741679 0.85 TRPV3 (0.41) CYP2D6HRH1TRPV3KCNH2CHRM1
SCHEMBL740324 0.84 CYP2C9 (0.44) CYP2D6HRH1TRPV3KCNH2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed