SCHEMBL740966

SCHEMBL740966

COCCCn1c(C2CCCN(C(=O)O)C2)nc2cc(C)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.44
HRH1 P35367 2/20 0.44
CYP2D6 P10635 1/20 0.44
P2RX3 P56373 3/20 0.44
P2RX2 Q9UBL9 1/20 0.44
CHRM1 P11229 1/20 0.43
JAK2 O60674 4/20 0.41
JAK1 P23458 4/20 0.41
TYK2 P29597 4/20 0.41
JAK3 P52333 4/20 0.41
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
ADORA2A P29274 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
PROKR1 Q8TCW9 2/20 0.40
CNR2 P34972 1/20 0.39
USP2 O75604 1/20 0.39
POLB P06746 1/20 0.39
ITK Q08881 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL765031 0.88 P2RX3 (0.45) KCNH2HRH1CYP2D6P2RX3P2RX2
SCHEMBL739857 0.87 HRH1 (0.57) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL740730 0.84 HRH1 (0.44) KCNH2HRH1CYP2D6CHRM1ADORA2A
SCHEMBL739392 0.84 KCNH2 (0.45) KCNH2HRH1CYP2D6CHRM1HCRTR1
SCHEMBL739667 0.84 KCNH2 (0.43) KCNH2HRH1CYP2D6CHRM1ADORA2A
SCHEMBL741439 0.83 HRH1 (0.46) KCNH2HRH1CYP2D6CHRM1PROKR1
SCHEMBL740454 0.82 ADORA2A (0.51) KCNH2HRH1CYP2D6CHRM1ADORA2A
SCHEMBL740553 0.80 KCNH2 (0.39) KCNH2HRH1CYP2D6P2RX3P2RX2
SCHEMBL740554 0.80 KCNH2 (0.39) KCNH2HRH1CYP2D6P2RX3P2RX2
SCHEMBL762833 0.79 POLB (0.43) KCNH2HRH1CYP2D6P2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed