SCHEMBL7407489

SCHEMBL7407489

CCCC[N+](C)(C)CCCCNC(=O)CN1CCC(C(=O)O)C1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR5 Q9H228 7/20 0.42
S1PR4 O95977 1/20 0.42
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42
GNAI3 P08754 2/20 0.41
GNAO1 P09471 2/20 0.41
GNAI1 P63096 2/20 0.41
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
NAAA Q02083 1/20 0.35
GAA P10253 2/20 0.34
BCHE P06276 1/20 0.34
KDM4E B2RXH2 2/20 0.34
POLB P06746 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
OPRD1 P41143 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7522334 0.89 S1PR5 (0.48) S1PR5S1PR4S1PR1S1PR3GNAI3
SCHEMBL8784235 0.83 S1PR5 (0.44) S1PR5S1PR4S1PR1S1PR3GNAI3
SCHEMBL13343830 0.71 BCHE (0.66) GNAI3GNAO1GNAI1ALDH1A1SIGMAR1
SCHEMBL14554075 0.70 S1PR5 (0.56) S1PR5S1PR4S1PR1S1PR3SMN1; SMN2
SCHEMBL13766174 0.70 S1PR5 (0.56) S1PR5S1PR4S1PR1S1PR3SMN1; SMN2
SCHEMBL7512062 0.69 S1PR5 (0.57) S1PR5S1PR4S1PR1S1PR3SMN1; SMN2
SCHEMBL7402269 0.69 SIGMAR1 (0.54) S1PR5S1PR4S1PR1S1PR3ALDH1A1
SCHEMBL6897984 0.68 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2SIGMAR1NAAAKDM4E
SCHEMBL7398353 0.68 GAA (0.45) S1PR5S1PR4S1PR1S1PR3ALDH1A1
SCHEMBL7508959 0.68 S1PR5 (0.56) S1PR5S1PR4S1PR1S1PR3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003740-A2 PYRROLIDINE-3-CARBOXYLIC ACID DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGOISTS Abbott Laboratories (US) 2000-05-31 EP disclosed
WO-1999006397-A2 PYRROLIDINE-3-CARBOXYLIC ACID DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGONISTS ABBOTT LABORATORIES (US) 1999-02-11 WO disclosed
EP-0885215-A1 NOVEL BENZO-1,3-DIOXOLYL- AND BENZOFURANYL SUBSTITUTED PYRROLIDINE DERIVATIVES AS ENDOTHELIN ANTAGONISTS Abbott Laboratories (US) 1998-12-23 EP disclosed
WO-1997030045-A1 NOVEL BENZO-1,3-DIOXOLYL- AND BENZOFURANYL SUBSTITUTED PYRROLIDINE DERIVATIVES AS ENDOTHELIN ANTAGONISTS ABBOTT LABORATORIES (US) 1997-08-21 WO disclosed