SCHEMBL7408015

SCHEMBL7408015

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2cc(Cl)ccc2Cl)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 1/20 0.38
HTT P42858 1/20 0.37
ITGB3 P05106 6/20 0.36
ITGA2B P08514 5/20 0.36
AR P10275 1/20 0.35
ITGB1 P05556 1/20 0.35
ITGA5 P08648 1/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
MMP1 P03956 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP8 P22894 1/20 0.34
PPARG P37231 2/20 0.33
BCL2 P10415 1/20 0.33
F2 P00734 4/20 0.33
TMPRSS6 Q8IU80 4/20 0.33
PPARA Q07869 1/20 0.33
ITGAV P06756 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416348 0.94 ITGB3 (0.36) ITGB3ITGA2BITGB1ITGA5CNR1
SCHEMBL7414111 0.92 PPARD (0.39) HTTITGB3ITGA2BITGB1ITGA5
SCHEMBL7414232 0.92 ITGB3 (0.37) HTTITGB3ITGA2BITGB1ITGA5
SCHEMBL7418892 0.91 CYP3A4 (0.43) HTTITGB3ITGA2BITGB1ITGA5
SCHEMBL7412118 0.91 ACLY (0.38) ITGB3ITGA2BITGB1ITGA5F2
SCHEMBL7415119 0.90 ITGB1 (0.39) HTTITGB3ITGA2BITGB1ITGA5
SCHEMBL7416127 0.90 ITGB3 (0.37) HTTITGB3ITGA2BITGB1ITGA5
Trifluoroacetic Acid SCHEMBL7408006 0.90 HTT (0.46) PSMB5HTTITGB3ITGA2BAR
SCHEMBL7415220 0.89 ITGB1 (0.36) ITGB3ITGA2BITGB1ITGA5PPARG
SCHEMBL7414434 0.89 F2 (0.42) HTTITGB3ITGA2BMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed