SCHEMBL7414232

SCHEMBL7414232

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2cc(Cl)c(Cl)cc2Cl)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.37
ITGA2B P08514 9/20 0.37
ITGB1 P05556 1/20 0.36
ITGA5 P08648 1/20 0.36
HTT P42858 1/20 0.34
F2 P00734 4/20 0.34
TMPRSS6 Q8IU80 4/20 0.34
PPARA Q07869 4/20 0.34
PPARD Q03181 2/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416348 0.92 ITGB3 (0.36) ITGB3ITGA2BITGB1ITGA5F2
SCHEMBL7408015 0.92 PSMB5 (0.38) ITGB3ITGA2BITGB1ITGA5HTT
SCHEMBL7418101 0.91 PPARD (0.41) ITGB3ITGA2BITGB1ITGA5PPARA
SCHEMBL7414111 0.91 PPARD (0.39) ITGB3ITGA2BITGB1ITGA5HTT
SCHEMBL7415119 0.90 ITGB1 (0.39) ITGB3ITGA2BITGB1ITGA5HTT
SCHEMBL7416127 0.89 ITGB3 (0.37) ITGB3ITGA2BITGB1ITGA5HTT
SCHEMBL7415413 0.89 TMPRSS6 (0.38) ITGB3ITGA2BITGB1ITGA5F2
Trifluoroacetic Acid SCHEMBL7414224 0.89 ITGB3 (0.47) ITGB3ITGA2BITGB1ITGA5HTT
SCHEMBL7408394 0.89 ITGB3 (0.37) ITGB3ITGA2BITGB1ITGA5F2
SCHEMBL7412118 0.89 ACLY (0.38) ITGB3ITGA2BITGB1ITGA5F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed