SCHEMBL7416348

SCHEMBL7416348

N=C(N)NOCCCOc1ccc(C[C@H](NS(=O)(=O)c2ccc(Cl)cc2Cl)C(=O)OC(=O)C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.36
ITGA2B P08514 7/20 0.36
ITGB1 P05556 1/20 0.35
ITGA5 P08648 1/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
TRPV4 Q9HBA0 2/20 0.34
ITGAV P06756 2/20 0.34
F2 P00734 4/20 0.33
TMPRSS6 Q8IU80 4/20 0.33
PPARA Q07869 1/20 0.33
RHOC P08134 1/20 0.32
RHOA P61586 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7408015 0.94 PSMB5 (0.38) ITGB3ITGA2BITGB1ITGA5CNR1
SCHEMBL7418101 0.92 PPARD (0.41) ITGB3ITGA2BITGB1ITGA5TRPV4
SCHEMBL7414232 0.92 ITGB3 (0.37) ITGB3ITGA2BITGB1ITGA5F2
SCHEMBL7412118 0.91 ACLY (0.38) ITGB3ITGA2BITGB1ITGA5F2
SCHEMBL7415220 0.90 ITGB1 (0.36) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7415119 0.90 ITGB1 (0.39) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7416127 0.90 ITGB3 (0.37) ITGB3ITGA2BITGB1ITGA5F2
Trifluoroacetic Acid SCHEMBL7416343 0.90 ITGB3 (0.46) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7418892 0.89 CYP3A4 (0.43) ITGB3ITGA2BITGB1ITGA5ITGAV
SCHEMBL7414434 0.89 F2 (0.42) ITGB3ITGA2BF2TMPRSS6RHOC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed