SCHEMBL7409113

SCHEMBL7409113

[AsH2]c1cccc(-c2ccc(OCCN3CCCC3)c3ccccc23)n1

nearest known ligand 0.75

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 8/20 0.75
NOS1 P29475 8/20 0.75
NOS2 P35228 8/20 0.75
TDP1 Q9NUW8 2/20 0.50
HRH3 Q9Y5N1 4/20 0.48
HTR2A P28223 2/20 0.48
HTR7 P34969 2/20 0.48
HTR6 P50406 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5834017 0.86 NOS3 (1.00) NOS3NOS1NOS2TDP1HRH3
SCHEMBL5833909 0.85 NOS3 (0.98) NOS3NOS1NOS2TDP1HRH3
SCHEMBL7083997 0.79 NOS3 (0.85) NOS3NOS1NOS2TDP1HRH3
SCHEMBL5834368 0.77 NOS3 (1.00) NOS3NOS1NOS2
SCHEMBL7126075 0.76 NOS3 (0.79) NOS3NOS1NOS2HRH3HTR2A
SCHEMBL5833641 0.76 NOS3 (0.81) NOS3NOS1NOS2
SCHEMBL7126072 0.76 NOS3 (0.60) NOS3NOS1NOS2HRH3HTR2A
SCHEMBL5833437 0.74 NOS1 (0.78) NOS3NOS1NOS2HTR2AHTR7
SCHEMBL14970486 0.74 HRH3 (0.81) NOS3NOS1NOS2TDP1HRH3
SCHEMBL5833259 0.73 NOS3 (0.75) NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1007520-A1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NOS INHIBITORS Pfizer Products Inc. (US) 2000-06-14 EP disclosed
WO-1999010339-A1 2-AMINOPYRIDINES CONTAINING FUSED RING SUBSTITUENTS AS NOS INHIBITORS PFIZER PRODUCTS INC. (US) 1999-03-04 WO disclosed