SCHEMBL7409358

SCHEMBL7409358

Fc1ccc(NC(c2cccc(OC(F)(F)F)c2)C2CCN(CCCOc3ccccc3)C2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.41
HTR1A P08908 3/20 0.41
DRD2 P14416 2/20 0.41
HTR7 P34969 2/20 0.41
HTR6 P50406 1/20 0.41
TMEM97 Q5BJF2 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
HTR2A P28223 1/20 0.39
HRH1 P35367 1/20 0.39
DRD3 P35462 1/20 0.39
KCNH2 Q12809 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
CACNA1B Q00975 2/20 0.38
CASR P41180 1/20 0.38
BCHE P06276 1/20 0.38
SLC6A3 Q01959 1/20 0.38
CCR2 P41597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7412531 0.87 DRD2 (0.47) HTR1ADRD2HTR7HTR6TMEM97
SCHEMBL7418258 0.82 HRH3 (0.46) HTR1ADRD2HTR7HTR6TMEM97
SCHEMBL7410875 0.81 DRD2 (0.50) HTR1ADRD2HTR7TMEM97SIGMAR1
Hydrochloric Acid SCHEMBL7413702 0.80 DRD2 (0.48) HTR1ADRD2HTR7TMEM97SIGMAR1
Hydrochloric Acid SCHEMBL7413705 0.80 DRD2 (0.48) HTR1ADRD2HTR7TMEM97SIGMAR1
SCHEMBL7407159 0.79 DRD2 (0.47) EPHX2HTR1ADRD2HTR7TMEM97
SCHEMBL7415382 0.77 DRD2 (0.47) EPHX2HTR1ADRD2HTR7TMEM97
SCHEMBL7415518 0.73 UBE2M (0.49) SIGMAR1BCHESLC6A3CCR2
SCHEMBL10560937 0.72 HTR2A (0.55) HTR1ADRD2HTR7TMEM97SIGMAR1
SCHEMBL7413539 0.71 DRD2 (0.51) HTR1ADRD2HTR7TMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5198449-A N-substituted alpha-arylazacycloalkylmethanamines and their use as cardiovascular agents A. H. ROBINS COMPANY INCORPORATED (US) 1993-03-30 US disclosed