SCHEMBL7409504

SCHEMBL7409504

NCc1cccc(Nc2[c]cccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.44
BPTF Q12830 1/20 0.41
LOXL2 Q9Y4K0 3/20 0.41
BRD4 O60885 1/20 0.38
PNMT P11086 1/20 0.38
ENPP2 Q13822 1/20 0.38
CFD P00746 4/20 0.38
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
SYK P43405 1/20 0.35
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
AR P10275 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
SIRT1 Q96EB6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7405571 0.84 TOP2A (0.49) ENPP2SYKMEN1ALDH1A1AR
SCHEMBL27903338 0.78 HTR6 (0.53) HTR6BPTFLOXL2BRD4PNMT
SCHEMBL27473567 0.77 ALDH1A1 (0.60) HTR6BPTFLOXL2BRD4PNMT
SCHEMBL27982990 0.75 SIRT1 (0.53) HTR6BPTFLOXL2BRD4PNMT
SCHEMBL693995 0.75 RAPGEF4 (0.45) MEN1ALDH1A1ARMAPTKMT2A
SCHEMBL72023 0.74 HSD17B10 (0.50) MEN1ALDH1A1ARMAPTKMT2A
SCHEMBL8725838 0.74 EGFR (0.39) MEN1ALDH1A1ARMAPTKMT2A
Biphenyl SCHEMBL27570267 0.73 TAAR1 (0.55) HTR6LOXL2PNMTENPP2CFD
SCHEMBL6986651 0.71 MEN1 (0.53) MEN1ALDH1A1MAPTKMT2A
SCHEMBL693983 0.71 IDH2 (0.54) MEN1ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948525-A1 CYCLIC PEPTIDE DERIVATIVES MERCK PATENT GmbH (DE) 1999-10-13 EP disclosed
WO-1998027112-A1 CYCLIC PEPTIDE DERIVATIVES MERCK PATENT GMBH (DE) 1998-06-25 WO disclosed