SCHEMBL762833

SCHEMBL762833

CCCCn1c([C@@H]2CCCN(C(=O)OC(C)(C)C)C2)nc2cc(C)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.43
P2RX3 P56373 2/20 0.42
P2RX2 Q9UBL9 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
HPGD P15428 1/20 0.41
RECQL P46063 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CNR2 P34972 1/20 0.41
TLR8 Q9NR97 1/20 0.41
KCNH2 Q12809 2/20 0.40
PROKR1 Q8TCW9 2/20 0.40
HPGDS O60760 1/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
TRPV3 Q8NET8 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL765031 0.91 P2RX3 (0.45) P2RX3P2RX2KDM4EALDH1A1GLA
SCHEMBL26263181 0.84 KDM4E (0.40) POLBP2RX3P2RX2KDM4EALDH1A1
SCHEMBL740716 0.82 CYP2D6 (0.41) P2RX3P2RX2KCNH2HPGDSTRPV3
SCHEMBL740717 0.82 CYP2D6 (0.41) P2RX3P2RX2KCNH2HPGDSTRPV3
SCHEMBL762854 0.80 P2RX7 (0.42) POLBALDH1A1KCNH2HPGDSJAK2
SCHEMBL762590 0.80 P2RX7 (0.42) POLBALDH1A1HPGDCNR2KCNH2
SCHEMBL741975 0.79 KCNH2 (0.52) POLBKCNH2HPGDSCYP2D6HRH1
SCHEMBL741974 0.79 KCNH2 (0.52) POLBKCNH2HPGDSCYP2D6HRH1
SCHEMBL762531 0.79 TLR8 (0.44) CNR2TLR8HPGDSTP53
SCHEMBL740966 0.79 KCNH2 (0.44) POLBP2RX3P2RX2CNR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed